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Serotonin 2B receptor is required for heart development

Canan G Nebigil , D.-S. Choi , André Dierich , Pierre Hickel , Marianne Le Meur , et al.
Proceedings of the National Academy of Sciences of the United States of America, 2000, 97 (17), pp.9508-9513. ⟨10.1073/pnas.97.17.9508⟩
Article dans une revue hal-02926424v1
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Oxidative Metabolism of Ferrocene Analogues of Tamoxifen: Characterization and Antiproliferative Activities of the Metabolites

Marie-Aude Richard , Didier Hamels , Pascal Pigeon , Siden Top , Patrick M. Dansette , et al.
ChemMedChem, 2015, 10 (6), pp.981-990. ⟨10.1002/cmdc.201500075⟩
Article dans une revue hal-01230370v1
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Specific effect of a dopamine partial agonist on counterfactual learning: evidence from Gilles de la Tourette syndrome

Alexandre Salvador , Yulia Worbe , Cécile Delorme , Giorgio Coricelli , Raphaël Gaillard , et al.
Scientific Reports, 2017, 7, pp.6292. ⟨10.1038/s41598-017-06547-8⟩
Article dans une revue hal-01580171v1
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Les analogues de l'apéline métaboliquement stables dans le traitement de l'hyponatrémie et de l'insuffisance cardiaque après infarctus du myocarde

Pierre-Emmanuel Girault-Sotias
Pharmacologie. Université Paris Cité, 2022. Français. ⟨NNT : 2022UNIP5006⟩
Thèse tel-03986345v1
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LIT01-196, a Metabolically Stable Apelin-17 Analog, Normalizes Blood Pressure in Hypertensive DOCA-Salt Rats via a NO Synthase-dependent Mechanism

Adrien Flahault , Mathilde Keck , Pierre-Emmanuel Girault-Sotias , Lucie Esteoulle , Nadia de Mota , et al.
Frontiers in Pharmacology, 2021, 12, ⟨10.3389/fphar.2021.715095⟩
Article dans une revue hal-03322968v1
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QGC606: A Best-in-Class Orally Active Centrally Acting Aminopeptidase A Inhibitor Prodrug for Treating Heart Failure Following Myocardial Infarction

Solène E Boitard , Mathilde Keck , Robin Deloux , Pierre-Emmanuel Girault-Sotias , Yannick Marc , et al.
Canadian Journal of Cardiology, 2022, 38 (6), pp.815-827. ⟨10.1016/j.cjca.2022.01.019⟩
Article dans une revue hal-03834295v1
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A Curvilinear-Path Umbrella Sampling Approach to Characterizing the Interactions Between Rapamycin and Three FKBP12 Variants

Dhananjay C Joshi , Charlie Gosse , Shu-Yu Huang , Jung-Hsin Lin
Frontiers in Molecular Biosciences, 2022, 9, pp.879000. ⟨10.3389/fmolb.2022.879000⟩
Article dans une revue hal-03845982v1
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Identification and pharmacological properties of E339–3D6, the first nonpeptidic apelin receptor agonist

Xavier Itturioz , Rodrigo Alvear-Perez , Nadia de Mota , Christel Franchet , Fabrice Guillier , et al.
FASEB Journal, 2010, ⟨10.1096/fj.09-140715⟩
Article dans une revue hal-02196074v1
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Optical control of neuronal ion channels and receptors

Pierre Paoletti , Graham Ellis-Davies , Alexandre Mourot
Nature Reviews Neuroscience, 2019, 20 (9), pp.514-532. ⟨10.1038/s41583-019-0197-2⟩
Article dans une revue hal-02352284v1

Protective effect of the octadecaneuropeptide on hydrogen peroxide-induced oxidative stress and cell death in cultured rat astrocytes

Yosra Hamdi , Olfa Masmoudi-Kouki , Hadhemi Kaddour , Feten Belhadj , Pierrick Gandolfo , et al.
Journal of Neurochemistry, 2011, 118 (3), pp.416-428. ⟨10.1111/j.1471-4159.2011.07315.x⟩
Article dans une revue hal-01962753v1

Identification of 26RFa, a hypothalamic neuropeptide of the RFamide peptide family with orexigenic activity

Nicolas Chartrel , Cynthia Dujardin , Youssef Anouar , Jérôme Leprince , Annick Decker , et al.
Proceedings of the National Academy of Sciences of the United States of America, 2011, 100 (25), pp.15247-15252. ⟨10.1073/pnas.2434676100⟩
Article dans une revue hal-01960798v1
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Fonctionnement des récepteurs-canaux du glutamate

Marc Gielen
Médecine/Sciences, 2010, 26 (1), pp.67-72. ⟨10.1051/medsci/201026165⟩
Article dans une revue hal-01145444v1
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Astroglial Connexins Inactivation Increases Relapse of Depressive-like Phenotype after Antidepressant Withdrawal

Benjamin Portal , Flora Vasile , Jonathan Zapata , Camille Lejards , Abd El Kader Ait Tayeb , et al.
International Journal of Molecular Sciences, 2022, 23 (21), pp.13227. ⟨10.3390/ijms232113227⟩
Article dans une revue hal-04083321v1
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Activating the apelin receptor with LIT01-196, a metabolically stable apelin analog, reverses AVP-induced antidiuresis and hyponatremia

Adrien Flahault , Pierre-Emmanuel Girault-Sotias , Mathilde Keck , Rodrigo Alvear-Perez , Nadia de Mota , et al.
Nature Communications, 2021, 12 (1), ⟨10.1038/s41467-020-20560-y⟩
Article dans une revue hal-03285794v1

Treatment of inherited protein C deficiency by replacement therapy with the French purified plasma-derived protein C concentrate (PROTEXEL).

M. Dreyfus , A. Ladouzi , H. Chambost , Y. Gruel , B. Tardy , et al.
Vox Sanguinis, 2007, 93 (3), pp.233-40. ⟨10.1111/j.1423-0410.2007.00953.x⟩
Article dans une revue istex ujm-00440305v1
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Molecular Mechanism of Action of 2-Ferrocenyl-1,1-diphenylbut-1-ene on HL-60 Leukemia Cells

Alane Cabral De Oliveira , Emanuella Gomes Da Silva , Danilo Damasceno Rocha , Elisabeth A. Hillard , Pascal Pigeon , et al.
ChemMedChem, 2014, 9 (11), pp.2580-2586. ⟨10.1002/cmdc.201402219⟩
Article dans une revue istex hal-01230375v1
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Les oeuvres pharmacologiques de Galien dans l’enseignement, l’édition et la pratique de la médecine en France au seizième siècle

Daniel Béguin
Armelle Debru. Galen On Pharmacology. Philosophy, History and Medicine, Proceedings of the Vth International Galen Colloquium,, 16, Brill, pp.283-300, 1997, Studies in Ancient Medicine, 978-90-04-10403-7. ⟨10.1163/9789004377431_014⟩
Chapitre d'ouvrage hal-03177651v1
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Enhanced and preferential internalization of lipid nanocapsules into human glioblastoma cells: effect of a surface-functionalizing NFL peptide

Reatul Karim , Elise Lepeltier , Lucille Esnault , Pascal Pigeon , Laurent Lemaire , et al.
Nanoscale, 2018, 10, pp.13485-13501. ⟨10.1039/C8NR02132E⟩
Article dans une revue hal-01817763v1
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Brain renin-angiotensin system blockade with orally active aminopeptidase A inhibitor prevents cardiac dysfunction after myocardial infarction in mice

Solène Emmanuelle Boitard , Yannick Marc , Mathilde Keck , Nathalie Mougenot , Onnik Agbulut , et al.
Journal of Molecular and Cellular Cardiology, 2019, 127, pp.215-222. ⟨10.1016/j.yjmcc.2018.12.008⟩
Article dans une revue hal-02265448v1
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Allosteric regulation in NMDA receptors revealed by the genetically encoded photo-cross- linkers

Meilin Tian , Shixin Ye
Scientific Reports, 2016, 6, pp.34751. ⟨10.1038/srep34751⟩
Article dans une revue hal-01390600v1
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The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells

Rosamaria Lappano , Christophe Mallet , Bruno Rizzuti , Fedora Grande , Giulia Raffaella Galli , et al.
Cells, 2019, Molecular and Cellular Mechanisms of Cancers: Breast Cancer, 8 (6), pp.590. ⟨10.3390/cells8060590⟩
Article dans une revue hal-02273130v1
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Molecular, Structural, Functional, and Pharmacological Sites for Vesicular Glutamate Transporter Regulation

Nicolas Pietrancosta , Mahamadou Djibo , Stephanie Daumas , Salah El Mestikawy , Jeffrey D. Erickson
Molecular Neurobiology, 2020, 57 (7), pp.3118-3142. ⟨10.1007/s12035-020-01912-7⟩
Article dans une revue hal-03007881v1
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Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition

Simon Hayek , Nicolas Pietrancosta , Anna Hovhannisyan , Rodolphe Alves de Sousa , Nassima Bekaddour , et al.
European Journal of Medicinal Chemistry, 2020, 186, pp.111855. ⟨10.1016/j.ejmech.2019.111855⟩
Article dans une revue hal-02372490v1
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Antitumor Activity and Mechanism of Action of Hormonotoxin, an LHRH Analog Conjugated to Dermaseptin-B2, a Multifunctional Antimicrobial Peptide

Mickael Couty , Marie Dusaud , Micka Miro-Padovani , Liuhui Zhan , Patricia Zadigue , et al.
International Journal of Molecular Sciences, 2021, 22 (21), pp.11303. ⟨10.3390/ijms222111303⟩
Article dans une revue hal-03388092v1
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Quantifying the relationship between SARS-CoV-2 viral load and infectiousness

Aurélien Marc , Marion Kerioui , Julie Bertrand , François Blanquart , Oriol Mitjà , et al.
eLife, 2021, 10, ⟨10.7554/eLife.69302⟩
Article dans une revue hal-03405884v1

The octadecaneuropeptide ODN prevents 6-hydroxydopamine-induced apoptosis of cerebellar granule neurons through a PKC-MAPK-dependent pathway

Hadhemi Kaddour , Yosra Hamdi , David Vaudry , Magalie Basille , Laurence Desrues , et al.
Journal of Neurochemistry, 2013, 125 (4), pp.620-633. ⟨10.1111/jnc.12140⟩
Article dans une revue hal-01962763v1

Functional Characterization and Potential Applications for Enhanced Green Fluorescent Protein-and Epitope-Fused Human M1 Muscarinic Receptors

Maurice Chasserot-Golaz , Brigitte Goeldner , Claire O. Weill , Jean-Luc Galzi , Sylvette Chasserot-Golaz , et al.
Journal of Neurochemistry, 1999, 73 (2), pp.791-801. ⟨10.1046/j.1471-4159.1999.0730791.x⟩
Article dans une revue hal-02194329v1

Monitoring In Vivo Performances of Protein–Drug Conjugates Using Site-Selective Dual Radiolabeling and Ex Vivo Digital Imaging

Héloïse Cahuzac , Antoine Sallustrau , Carole Malgorn , Fabrice Beau , Peggy Barbe , et al.
Journal of Medicinal Chemistry, 2022, 65 (9), pp.6953 - 6968. ⟨10.1021/acs.jmedchem.2c00401⟩
Article dans une revue cea-03834302v1
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Connexin and pannexin hemichannels in brain glial cells: properties, pharmacology, and roles

Christian Giaume , Luc Leybaert , Christian C. Naus , Juan C. Sáez
Frontiers in Pharmacology, 2013, 4, pp.88. ⟨10.3389/fphar.2013.00088⟩
Article dans une revue hal-01578556v1
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Risk of early neurodevelopmental disorders associated with in utero exposure to valproate and other antiepileptic drugs: a nationwide cohort study in France

Joël Coste , Pierre-Olivier Blotiere , Sara Miranda , Yann Mikaeloff , Hugo Peyre , et al.
Scientific Reports, 2020, 10, pp.17362. ⟨10.1038/s41598-020-74409-x⟩
Article dans une revue hal-02976092v1